Relispa (40mg) 20 Tablets

Drotaverine 40mg Tablet primarily exerts its therapeutic effects through its action as a spasmolytic agent. It selectively inhibits phosphodiesterase type IV, leading to increased levels of cyclic adenosine monophosphate (cAMP) in smooth muscle cells. This rise in cAMP reduces calcium influx into the cells, thereby relaxing the smooth muscles and alleviating spasms. By targeting this specific enzyme, drotaverine effectively relaxes smooth muscle contractions without impacting normal gastrointestinal motility, making it a valuable medication for managing various conditions characterized by smooth muscle spasms.

Drotaverine 40mg

Spasmolytic (antispasmodic) agent.

Tablet

The following are the uses of Drotaverine 40mg Tablet:

• Used for relaxing smooth muscles and relieving painful muscle spasms in the abdomen, intestines, and urinary tract.
• Used to treat painful menstrual periods and pelvic pain in women.
• Used to manage pain and discomfort during kidney or bladder stones.
• Used to reduce inflammation and pain in the digestive tract caused by conditions like irritable bowel syndrome.
• Used for managing post-operative pain and discomfort.
• Used to alleviate pain and stiffness in conditions like fibromyalgia.
• Used to provide relief from muscle spasms and pain associated with musculoskeletal injuries.

Follow these dosage instructions:

• Adult Dosage

The recommended daily dosage is 40mg. The maximum dose is 80mg/daily.

• Child Dosage

The child's dosage is 20mg daily orally.

In the case of an overdose of Drotaverine 40mg Tablets, symptoms may include severe dizziness, fainting, rapid heartbeat, and in extreme cases, seizures. If you suspect an overdose, it is important to seek medical advice promptly. Do not induce vomiting, as this may worsen the situation. Medical professionals should be contacted immediately to provide appropriate treatment and support, which may include monitoring vital signs and providing symptomatic relief.

In the case of a missed dose of Drotaverine 40mg Tablet, it is important to take the missed dose as soon as you remember. However, if it is almost time for your next scheduled dose, skip the missed one. Never double the dose to make up for a missed one, as this may increase the risk of side effects. If you miss multiple doses, contact your healthcare provider for guidance on how to safely adjust your dosing schedule. It is advisable to set reminders or alarms to help you remember to take your medication on time to ensure the best treatment outcome.

To take Drotaverine 40mg Tablet, swallow the tablet whole with a glass of water, preferably with or after a meal, as directed by your healthcare professional.

Here are the conditions and situations when Drotaverine 40mg Tablet should not be taken:

• Avoid if allergic to Drotaverine or any similar medications.
• Not suitable for individuals with gastrointestinal bleeding.
• Contraindicated in patients with severe heart disease.
• Should not be used during active ulcerative colitis.
• Not recommended for individuals with kidney impairment or severe kidney disease.
• Avoid if you have a blockage in your intestines.
• Do not use if you have a history of hypersensitivity reactions to similar drugs.

The side effects of Drotaverine 40mg Tablet may include:

• Dry mouth
• Nausea and vomiting
• Diarrhea
• Dizziness
• Headache
• Skin rashes or itching
• Allergic reactions (rare)
• Cardiovascular issues (rare)

Following are the precautions and warnings for Drotaverine 40mg Tablet:

• This medication should not be taken if you are allergic to Drotaverine or any other similar antispasmodic drugs.
• Patients with liver or kidney disease should use with caution and under medical supervision as dosage adjustments may be necessary.
• Avoid driving or operating heavy machinery as Drotaverine can cause dizziness and blurred vision.
• Alcohol consumption should be avoided as it may increase the risk of side effects.
• Drotaverine is not recommended for use in children under 12 years of age.
• Pregnant and breastfeeding women should consult their doctor before taking this medication as it may pass into breast milk.
• Do not exceed the prescribed dosage, as it may lead to severe adverse effects.

Following are the drug interactions for Drotaverine 40mg Tablet:

• It may interact with other antispasmodic medications, leading to increased side effects and potential toxicity.
• Avoid using Drotaverine with anticholinergic drugs, as it can cause severe constipation and urinary retention.
• Concomitant use with certain antidepressants (e.g., tricyclic antidepressants) may enhance their side effects, especially on the cardiovascular system.
• Drotaverine can potentially reduce the effectiveness of antacids and proton pump inhibitors when taken simultaneously.
• When combined with antihistamines, it may cause excessive drowsiness and impaired cognitive function.
• This medication may interact with certain antibiotics, affecting their absorption and efficacy.
• Caution is advised when using Drotaverine with drugs metabolized by the liver, as it may alter their metabolism and increase side effects.

Following are the food interactions for Drotaverine 40mg Tablet:

• Drotaverine may be taken with or without food, but it is generally recommended to take it with food to reduce the risk of gastrointestinal side effects like nausea.
• Grapefruit and grapefruit juice should be avoided as they can inhibit certain enzymes, potentially altering the metabolism of the drug and increasing the risk of side effects.
• Alcohol consumption should be limited or avoided as it can increase the risk of gastrointestinal issues and may also enhance the sedative effects of Drotaverine.
• Caffeinated beverages like coffee and tea may be reduced as caffeine can stimulate the central nervous system, potentially counteracting the calming effects of Drotaverine on smooth muscles.
• High-fat meals may delay the absorption of Drotaverine, so it is advisable to avoid excessive fatty foods to ensure optimal medication effectiveness.
• Dairy products like milk may be consumed, but some individuals may experience slight changes in drug absorption, especially if they have lactose intolerance or related digestive issues.
• Spicy foods should be consumed in moderation as they can potentially irritate the gastrointestinal tract, which may be more sensitive while taking Drotaverine.
• Staying well-hydrated by drinking adequate water is essential to maintain overall health and to support the optimal functioning of the medication.

Drotaverine 40mg Tablets should be stored in a cool and dry place, preferably at room temperature below 25°C (77°F). Keep the tablets in their original packaging, ensuring the container is tightly sealed to protect them from moisture and light. Avoid storing the medication in the bathroom or kitchen, as these areas may have high humidity or temperature fluctuations that can degrade the tablets. Do not use the tablets if they show signs of damage or discoloration. It is crucial to dispose of expired or unused tablets properly by following local guidelines for pharmaceutical waste disposal. Do not flush them down the toilet or discard them in regular household waste, as this may harm the environment. Keep the medication out of the sight and reach of children and pets to prevent accidental consumption.

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Following are the quick tips for Drotaverine 40mg Tablet:

• Consult your doctor before use, especially if you have liver or kidney issues.
• Take the tablet as directed by your physician for effective pain relief.
• Swallow the tablet whole with water; do not crush or chew.
• Avoid alcohol consumption while taking this medication.
• If you experience dizziness, refrain from driving or operating heavy machinery.
• Inform your doctor about all medications you are taking to prevent potential interactions.
• Store the tablets in a cool, dry place, away from direct sunlight.